Resultats - Síntesis Orgànica Estereoselectiva
Síntesis Orgànica Estereoselectiva
| Tesis Doctorals Dirigides / Theses |
| 2021 | 2022 | 2023 | 2024 | 2025 |
|---|
| Títol: Insights into Aminofluorination Strategies and Sphingosine Analogue Synthesis towards the Development of Selective SphK2 Inhibitors |
| Autor: Granell Fort, Albert |
| Director: Matheu Malpartida, María Isabel; Díaz Giménez, María Yolanda |
| Universitat: N/D |
| Any: 2024 |
| País: N/D |
| Títol: Targeting Des1: Syntheses of ceramide analogues with a rigid scaffold, inhibitory assays, and AF2-assisted structural insights reveal PR280 as a potent inhibitor |
| Autor: Rivero Prieto, Pablo |
| Director: Díaz Giménez, María Yolanda; Matheu Malpartida, María Isabel |
| Universitat: N/D |
| Any: 2024 |
| País: N/D |
| Títol: Reagents and methodologies for the introduction of thiofluoroalkyl and fluorosulfur motifs |
| Autor: Bernús Pérez, Miguel |
| Director: Boutureira Martín, Omar |
| Universitat: N/D |
| Any: 2023 |
| País: N/D |
| Títol: Stereoselective synthesis of fluorinated glycoconjugates.Tuning physicochemical parameters for therapeutic drug development |
| Autor: Bascuas Jiménez De Bagües, Isabel |
| Director: Boutureira Martín, Omar |
| Universitat: N/D |
| Any: 2022 |
| País: N/D |
| Publicacions en Revista / Papers |
| 2021 | 2022 | 2023 | 2024 | 2025 |
|---|
| Títol: Impact of Fluorine Pattern on Lipophilicity and Acid-Base Properties of 2-(Thiofluoroalkyl)pyridines: Insights from Experiments and Statistical Modeling |
| Autors: Bernús, M; Núñez, GD; Hartley, WC; Guasch, M; Mestre, J; Besora, M; Carbó, JJ; Boutureira, O |
| Any: 2025 Clau: Article |
| Revista: Journal Of Medicinal Chemistry |
| País: N/D |
| Títol: Syntheses of differentially fluorinated triazole-based 1-deoxysphingosine analogues en route to SphK inhibitors |
| Autors: Cardona, Adria; Ivanova, Varbina; Beltran-Debon, Raul; Barril, Xavier; Castillon, Sergio; Diaz, Yolanda; Matheu, M Isabel |
| Any: 2025 Clau: Article |
| Revista: Organic & Biomolecular Chemistry |
| País: N/D |
| Títol: Electrophilic glycoluril-based reagents for atom-economic thiocyanation and selenocyanation of (hetero)arenes |
| Autors: Casasús, P; Mestre, J; Radlowska, R; Bernús, M; Boutureira, O |
| Any: 2025 Clau: Article |
| Revista: Organic & Biomolecular Chemistry |
| País: N/D |
| Títol: Palladium-Catalyzed Telomerization of Isoprene with Amines: Ligands and Solvents Working Together to Improve the Selectivity |
| Autors: Colavida, J; Penido, RG; Collado, A; Ricart, JM; Godard, C; Claver, C; Carbó, JJ; dos Santos, EN; Castillon, S |
| Any: 2025 Clau: Article |
| Revista: Chemcatchem |
| País: N/D |
| Títol: meta-Selective thiofluoroalkylation of substituted pyridines via Zincke imines |
| Autors: Hartley, WC; Huerta, A; Negredo, JC; Boutureira, O |
| Any: 2025 Clau: Article |
| Revista: Organic Chemistry Frontiers |
| País: N/D |
| Títol: A modular flow platform for sulfur(VI) fluoride exchange ligation of small molecules, peptides and proteins |
| Autors: Bernús, M; Mazzarella, D; Stanic, J; Zhai, ZR; Yeste-Vázquez, A; Boutureira, O; Gargano, AFG; Grossmann, TN; Noël, T |
| Any: 2024 Clau: Article |
| Revista: Nature Synthesis |
| País: N/D |
| Títol: Need for therapeutic escalation in patients with refractory ulcerative proctitis: Results from the PROCU study of the ENEIDA registry |
| Autors: Ferreiro-Iglesias, R; Silva, SP; Marín, S; Casanova, MJ; Mañosa, M; González-Muñoza, C; de Francisco, R; Caballol, B; Arias, L; Piqueras, M; Zabana, Y; Rivero, M; Calvet, X; Mesonero, F; Trastoy, PV; Nistal, RB; Perosanz, RG; Vega, P; Gonzalez-Vivo, M; Iborra, M; Bermejo, F; Madero, L; Rodríguez-Lago, I; Gonzalez, MR; Vera, I; Díaz, AP; Vela, M; Medina, LT; Van Domselaar, M; Gomollón, F; Iglesias, E; Gisbert, JP; Calafat, M; Giordano, A; Pérez-Martínez, I; Ricart, E; Sicilia, B; Mena, R; Esteve, M; Rivas, C; Brunet-Mas, E; Fernández, C; Turrión, MAD; Jiménez, BV; Calvo, MQ; Expósito, CR; Márquez-Mosquera, L; Nos, P; Granja, A; Gutiérrez, A; Cabriada, JL; Cruz, DH; Calvo, M; Pérez, JP; Díaz, YR; Casal, DB; Menacho, M; Leal, C; Lucendo, AJ; Royo, V; Olivares, S; Herrero, BA; Carrillo-Palau, M; Alvarez, PG; Marcos, NM; Martínez-Pérez, TD; Villafranca, MCM; Almela, P; Argüelles-Arias, F; Legido, J; Coronel, AMF; Nieto, L; Domènech, E; Acosta, MBD |
| Any: 2024 Clau: Article |
| Revista: Alimentary Pharmacology & Therapeutics |
| País: N/D |
| Títol: In-Flow Generation of Thionyl Fluoride (SOF2) Enables the Rapid and Efficient Synthesis of Acyl Fluorides from Carboxylic Acids |
| Autors: Mazzarella, D; Stanic, J; Bernus, M; Mehdi, AS; Henderson, CJ; Boutureira, O; Noël, T |
| Any: 2024 Clau: Article |
| Revista: Jacs Au |
| País: N/D |
| Títol: Targeting dihydroceramide desaturase 1 (Des1): Syntheses of ceramide analogues with a rigid scaffold, inhibitory assays, and AlphaFold2-assisted structural insights reveal cyclopropenone PR280 as a potent inhibitor |
| Autors: Rivero, P; Ivanova, V; Barril, X; Casampere, M; Casas, J; Fabriàs, G; Díaz, Y; Matheu, MI |
| Any: 2024 Clau: Article |
| Revista: Bioorganic Chemistry |
| País: N/D |
| Títol: Tetrafluoroethylation of Electron-Rich Alkenyl Iodides Enabled by in situ Generation of Solvent-Stabilized "Ligandless" CuCF2CF2H |
| Autors: Segovia, CM; Porto, LLTN; Casasús, P; Bascuas, I; Ahmad, A; Mestre, J; Bernus, M; Castillón, S; Baker, RT; Boutureira, O |
| Any: 2024 Clau: Article |
| Revista: Advanced Synthesis & Catalysis |
| País: N/D |
| Títol: A unified flow strategy for the preparation and use of trifluoromethyl-heteroatom anions |
| Autors: Spennacchio, M; Bernús, M; Stanic, J; Mazzarella, D; Colella, M; Douglas, JJ; Boutureira, O; Noël, T |
| Any: 2024 Clau: Article |
| Revista: Science |
| País: N/D |
| Títol: Bench-Stable Electrophilic Reagents for the Direct Di- and Trifluoroethylthiolation of Indoles |
| Autors: Casasus, P; Mestre, J; Bernus, M; Castillon, S; Boutureira, O |
| Any: 2023 Clau: Article |
| Revista: Advanced Synthesis & Catalysis |
| País: N/D |
| Títol: Bringing Selectivity in H/D Exchange Reactions Catalyzed by Metal Nanoparticles through Modulation of the Metal and the Ligand Shell |
| Autors: Martinez-Espinar, F; Salom-Català, A; Bresó-Femenia, E; Claver, C; Baletto, F; Ricart, JM; Chaudret, B; Carbó, JJ; Godard, C; Castillon, S |
| Any: 2023 Clau: Article |
| Revista: Inorganic Chemistry |
| País: N/D |
| Títol: Stereoselective access to 2-deoxy-2-trifluoromethyl sugar mimetics by trifluoromethyl-directed 1,2-trans glycosylation |
| Autors: Mestre, J; Bascuas, I; Bernús, M; Castillón, S; Boutureira, O |
| Any: 2023 Clau: Article |
| Revista: Organic Chemistry Frontiers |
| País: N/D |
| Títol: Probing Site-Selective Conjugation Chemistries for the Construction of Homogeneous Synthetic Glycodendriproteins |
| Autors: Cobo, I; Matheu, MI; Castillón, S; Davis, BG; Boutureira, O |
| Any: 2022 Clau: Article |
| Revista: Chembiochem |
| País: N/D |
| Títol: Revealing 2-dimethylhydrazino-2-alkyl alkynyl sphingosine derivatives as sphingosine kinase 2 inhibitors: Some hints on the structural basis for selective inhibition |
| Autors: Corro-Moron, Macarena; Granell, Albert; Ivanova, Varbina; Domingo, Elena; Beltran-Debon, Raul; Barril, Xavier; Sanz, Maria-Jesus; Matheu, M Isabel; Castillon, Sergio; Diaz, Yolanda |
| Any: 2022 Clau: Article |
| Revista: Bioorganic Chemistry |
| País: N/D |
| Títol: Association between histological diaphragm atrophy and ultrasound diaphragm expiratory thickness in ventilated patients |
| Autors: Dot, Irene; Perez-Teran, Purificacion; Frances, Albert; Diaz, Yolanda; Vila-Vilardell, Clara; Salazar-Degracia, Anna; Chalela, Roberto; Barreiro, Esther; Rodriguez-Fuster, Alberto; Ramon Masclans, Joan; Marin-Corral, Judith |
| Any: 2022 Clau: Article |
| Revista: Journal Of Intensive Care |
| País: N/D |
| Títol: Electrophilic Reagents for the Direct Incorporation of Uncommon SCF2CF2H and SCF2CF3 Motifs |
| Autors: Mestre, J; Bernu, M; Castillon, S; Boutureira, O |
| Any: 2022 Clau: Article |
| Revista: Journal Of Organic Chemistry |
| País: N/D |
| Títol: New Co and Mn Catalysts Bearing ONO Ligands Containing Nucleophile for the Coupling of CO2 and Propylene Oxide |
| Autors: Viciano, M; Muñoz, BK; Zangrando, E; Godard, C; Castillón, S; González, MDB; García-Ruíz, M; Claver, C |
| Any: 2022 Clau: Article |
| Revista: Catalysts |
| País: N/D |
| Títol: Toward the stereoselective synthesis of zaragozic acid framework: A desilylation-aldol reaction approach |
| Autors: Kurniawan, YD; Tuck, KL; Castillón, S; Robinson, AJ |
| Any: 2021 Clau: Article |
| Revista: Tetrahedron Letters |
| País: N/D |
| Títol: Metal complexes bearing ONO ligands as highly active catalysts in carbon dioxide and epoxide coupling reactions |
| Autors: Munoz, BK; Viciano, M; Godard, C; Castillon, S; Garcia-Ruiz, M; Gonzalez, MDB; Claver, C |
| Any: 2021 Clau: Article |
| Revista: Inorganica Chimica Acta |
| País: N/D |
| Llibres / Books |
| 2021 | 2022 | 2023 | 2024 | 2025 |
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| Capítols de Llibre / Book chapters |
| 2021 | 2022 | 2023 | 2024 | 2025 |
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| Altres Documents / Other documents |
| 2021 | 2022 | 2023 | 2024 | 2025 |
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| Patents Sol.licitades / Patents |
| 2021 | 2022 | 2023 | 2024 | 2025 |
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| Congressos / Conferences |
| 2021 | 2022 | 2023 | 2024 | 2025 |
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